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Patch Drug Delivery allows for pharmaceuticals to be delivered across the skin
barrier and into systemic blood circulation. This type of delivery helps bypass
initial metabolism in the liver and the gastrointestinal tract that occurs with
oral medications.
Early transdermal drug delivery patches launched
in the 1980's were of a liquid reservoir type design. In this
configuration, the drug is dissolved in a liquid reservoir
vehicle, often alcohol based, which is separated from the skin
by a semi-permeable membrane and contact adhesive.
In the 1990's, technology improvements
led to the development of the matrix-type patch, which integrates
the active drug, skin permeability enhancer, and adhesive
into one "membrane-like" layer coated onto a flexible
protective backing film. The matrix system makes the patch
thinner, more comfortable, more discreet, provides for better
adhesion, and is less prone to causing skin irritation.(1)
In addition, matrix systems are not dependent upon the finite
volume of alcohol based liquid reservoirs and provide for
more consistent delivery of the drug over the dosing interval.(2)

(1) R.S. Berger, G.D. Cioppa, and C.O.
Dillard, Skin Tolerability and Adhesion Characteristics of
a New Matrix Patch and a Marketed Reservoir Patch for Estradiol
Delivery. Menopause. Vol. 4(1), 1997, 46-51.
(2) A.J. Bowen, V.A. John, M.E. Ramirez,
and W.R. Good, Bioavailability of Oestradiol from the AloraTM
(0.1 mg/day) Oestradiol Matrix Transdermal Delivery System
Compared with Estraderm® (0.1 mg/day). J Obstet &
Gynocol. Vol. 18(6), 1998, 577-582. |
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